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Design of a Hypoxia-Activated Prodrug Inhibitor of O(6)-Alkylguanine-DNA Alkyltransferase

The efficacy of agents that alkylate the O-6 position of guanine is inhibited by O(6)-alkylguanine-DNA alkyltransferase (AGT) which removes these lesions from the tumor DNA. To increase differential toxicity, inhibitors must selectively deplete AGT in tumors, while sparing normal tissues where this...

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Detalhes bibliográficos
Main Authors: Zhu, Rui, Seow, Helen A., Baumann, Raymond P., Ishiguro, Kimiko, Penketh, Philip G., Shyam, Krishnamurthy, Sartorelli, Alan C.
Formato: Artigo
Idioma:Inglês
Publicado em: 2012
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC3444633/
https://ncbi.nlm.nih.gov/pubmed/22932317
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmcl.2012.08.008
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