Lataa...

Extreme Entropy-Enthalpy Compensation in a Drug Resistant Variant of HIV-1 Protease

The development of HIV-1 protease inhibitors has been the historic paradigm of rational structure-based drug design, where structural and thermodynamic analyses have assisted in the discovery of novel inhibitors. While the total enthalpy and entropy change upon binding determine the affinity, often...

Täydet tiedot

Tallennettuna:
Bibliografiset tiedot
Päätekijät: King, Nancy M., Prabu-Jeyabalan, Moses, Bandaranayake, Rajintha M., Nalam, Madhavi N. L., Nalivaika, Ellen A., Özen, Ayşegül, Haliloglu, Türkan, Yılmaz, Neşe Kurt, Schiffer, Celia A.
Aineistotyyppi: Artigo
Kieli:Inglês
Julkaistu: 2012
Aiheet:
Linkit:https://ncbi.nlm.nih.gov/pmc/articles/PMC3594831/
https://ncbi.nlm.nih.gov/pubmed/22712830
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/cb300191k
Tagit: Lisää tagi
Ei tageja, Lisää ensimmäinen tagi!