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Structural analysis of bengamide derivatives as inhibitors of methionine aminopeptidases

Natural product-derived bengamides possess potent antiproliferative activity and target human methionine aminopeptidases (MetAPs) for their cellular effects. Several derivatives were designed, synthesized, and evaluated as MetAP inhibitors. Here, we present four new X-ray structures of human MetAP1...

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Enregistré dans:
Détails bibliographiques
Auteurs principaux: Xu, Wei, Lu, Jing-Ping, Ye, Qi-Zhuang
Format: Artigo
Langue:Inglês
Publié: 2012
Sujets:
Accès en ligne:https://ncbi.nlm.nih.gov/pmc/articles/PMC3470909/
https://ncbi.nlm.nih.gov/pubmed/22913487
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/jm3008695
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