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Structural analysis of bengamide derivatives as inhibitors of methionine aminopeptidases

Natural product-derived bengamides possess potent antiproliferative activity and target human methionine aminopeptidases (MetAPs) for their cellular effects. Several derivatives were designed, synthesized, and evaluated as MetAP inhibitors. Here, we present four new X-ray structures of human MetAP1...

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Библиографические подробности
Главные авторы: Xu, Wei, Lu, Jing-Ping, Ye, Qi-Zhuang
Формат: Artigo
Язык:Inglês
Опубликовано: 2012
Предметы:
Online-ссылка:https://ncbi.nlm.nih.gov/pmc/articles/PMC3470909/
https://ncbi.nlm.nih.gov/pubmed/22913487
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/jm3008695
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