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Structural analysis of inhibition of Mycobacterium tuberculosis methionine aminopeptidase by bengamide derivatives

Natural product-derived bengamides possess potent antiproliferative activity and target human methionine aminopeptidases for their cellular effects. Using bengamides as a template, several derivatives were designed and synthesized as inhibitors of methionine aminopeptidases of Mycobacterium tubercul...

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Autori principali: Lu, Jing-Ping, Yuan, Xiu-Hua, Ye, Qi-Zhuang
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2011
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC3365506/
https://ncbi.nlm.nih.gov/pubmed/22118830
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.ejmech.2011.11.017
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