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Cobicistat Boosts the Intestinal Absorption of Transport Substrates, Including HIV Protease Inhibitors and GS-7340, In Vitro

The experimental pharmacoenhancer cobicistat (COBI), a potent mechanism-based inhibitor of cytochrome P450 3A enzymes, was found to inhibit the intestinal efflux transporters P-glycoprotein and breast cancer resistance protein. Consistent with its transporter inhibition, COBI significantly increased...

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Bibliografiske detaljer
Main Authors: Lepist, Eve-Irene, Phan, Truc K., Roy, Anupma, Tong, Leah, MacLennan, Kelly, Murray, Bernard, Ray, Adrian S.
Format: Artigo
Sprog:Inglês
Udgivet: American Society for Microbiology 2012
Fag:
Online adgang:https://ncbi.nlm.nih.gov/pmc/articles/PMC3457391/
https://ncbi.nlm.nih.gov/pubmed/22850510
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1128/AAC.01089-12
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