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Synthesis and in vitro biological evaluation of carbonyl group-containing analogues for σ(1) receptors

To identify the ligands for σ(1) receptors that are potent and selective, the analogues of prezamicol and trozamicol scaffolds of carbonyl-containing vesicular acetylcholine transporter (VAChT) inhibitors were explored. Of the 23 analogues synthesized and tested, 5 displayed very high affinity for σ...

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Hlavní autoři: Wang, Wei, Cui, Jinquan, Lu, Xiaoxia, Padakanti, Prashanth K., Xu, Jinbin, Parsons, Stanley M., Luedtke, Robert R., Rath, Nigam P., Tu, Zhude
Médium: Artigo
Jazyk:Inglês
Vydáno: 2011
Témata:
On-line přístup:https://ncbi.nlm.nih.gov/pmc/articles/PMC3150604/
https://ncbi.nlm.nih.gov/pubmed/21732626
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/jm200203f
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