Inhibition of secreted phospholipases A(2) by 2-oxoamides based on α-amino acids: Synthesis, in vitro evaluation and molecular docking calculations

Lignende værker

• Development of a potent 2-oxoamide inhibitor of secreted phospholipase A(2) guided by molecular docking calculations and molecular dynamics simulations
  af: Vasilakaki, Sofia, et al.
  Udgivet: (2016)
• 2-Oxoamide inhibitors of cytosolic group IVA phospholipase A(2) with reduced lipophilicity
  af: Antonopoulou, Georgia, et al.
  Udgivet: (2016)
• 2-Oxoamides based on dipeptides as selective calcium-independent phospholipase A(2) inhibitors
  af: Smyrniotou, Anneta, et al.
  Udgivet: (2016)
• Binding Conformation of 2-Oxoamide Inhibitors to Group IVA Cytosolic Phospholipase A(2) Determined by Molecular Docking Combined with Molecular Dynamics
  af: Mouchlis, Varnavas D., et al.
  Udgivet: (2012)
• Structure-activity relationships of natural and non-natural amino acid-based amide and 2-oxoamide inhibitors of human phospholipase A(2) enzymes
  af: Antonopoulou, Georgia, et al.
  Udgivet: (2008)