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Discovery of Potent and Reversible Monoacylglycerol Lipase Inhibitors

Monoacylglycerol lipase (MGL) is a serine hydrolase involved in the biological deactivation of the endocannabinoid 2-arachidonoyl-sn-glycerol (2-AG). Previous efforts to design MGL inhibitors have focused on chemical scaffolds that irreversibly block the activity of this enzyme. Here, we describe tw...

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Dettagli Bibliografici
Autori principali: King, Alvin R., Dotsey, Emmanuel Y., Lodola, Alessio, Jung, Kwang Mook, Ghomian, Azar, Qiu, Yan, Fu, Jin, Mor, Marco, Piomelli, Daniele
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2009
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC3034734/
https://ncbi.nlm.nih.gov/pubmed/19875078
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.chembiol.2009.09.012
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