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Allosteric Interactions between the Myristate- and ATP-Site of the Abl Kinase

Abl kinase inhibitors targeting the ATP binding pocket are currently employed as potent anti-leukemogenic agents but drug resistance has become a significant clinical limitation. Recently, a compound that binds to the myristate pocket of Abl (GNF-5) was shown to act cooperatively with nilotinib, an...

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Hlavní autoři: Iacob, Roxana E., Zhang, Jianming, Gray, Nathanael S., Engen, John R.
Médium: Artigo
Jazyk:Inglês
Vydáno: Public Library of Science 2011
Témata:
On-line přístup:https://ncbi.nlm.nih.gov/pmc/articles/PMC3018526/
https://ncbi.nlm.nih.gov/pubmed/21264348
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1371/journal.pone.0015929
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