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Evaluation of Di-Sansalvamide A derivatives: Synthesis, structure-activity relationship, and mechanism of action

Described is the SAR of 18 Di-Sansalvamide A derivatives and the mechanism of action of the most potent compound. We show that this scaffold is a promising lead in the development of novel cancer therapeutics because it is: cytotoxic at nanomolar potency, inhibits a well-established oncogenic target...

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Hlavní autoři: Alexander, Leslie D., Sellers, Robert P., Davis, Melinda R., Ardi, Veronica C., Johnson, Victoria A., Vasko, Robert C., McAlpine, Shelli R.
Médium: Artigo
Jazyk:Inglês
Vydáno: 2009
Témata:
On-line přístup:https://ncbi.nlm.nih.gov/pmc/articles/PMC2805559/
https://ncbi.nlm.nih.gov/pubmed/20014866
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/jm901566c
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