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Transition state analogues in structures of ricin and saporin ribosome-inactivating proteins

Ricin A-chain (RTA) and saporin-L1 (SAP) catalyze adenosine depurination of 28S rRNA to inhibit protein synthesis and cause cell death. We present the crystal structures of RTA and SAP in complex with transition state analogue inhibitors. These tight-binding inhibitors mimic the sarcin–ricin recogni...

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Autors principals: Ho, Meng-Chiao, Sturm, Matthew B., Almo, Steven C., Schramm, Vern L.
Format: Artigo
Idioma:Inglês
Publicat: National Academy of Sciences 2009
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC2787146/
https://ncbi.nlm.nih.gov/pubmed/19920175
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1073/pnas.0911606106
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