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Affinity modulation of small-molecule ligands by borrowing endogenous protein surfaces

A general strategy is described for improving the binding properties of small-molecule ligands to protein targets. A bifunctional molecule is created by chemically linking a ligand of interest to another small molecule that binds tightly to a second protein. When the ligand of interest is presented...

Ausführliche Beschreibung

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Bibliographische Detailangaben
Hauptverfasser: Briesewitz, Roger, Ray, Gregory T., Wandless, Thomas J., Crabtree, Gerald R.
Format: Artigo
Sprache:Inglês
Veröffentlicht: The National Academy of Sciences 1999
Schlagworte:
Online Zugang:https://ncbi.nlm.nih.gov/pmc/articles/PMC26718/
https://ncbi.nlm.nih.gov/pubmed/10051576
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