Gold Catalysed Redox Synthesis of Imidazo[1,2-a]pyridine using Pyridine N-Oxide and Alkynes

由 Talbot, Eric P. A., Richardson, Melodie, McKenna, Jeffrey M., Toste, F. Dean
出版 2014

Chiral Diaryliodonium Phosphate Enables Light Driven Diastereoselective α-C(sp3)−H Acetalization

由 Ye, Baihua, Zhao, Jie, Zhao, Ke, McKenna, Jeffrey M., Toste, F. Dean
發表在 J Am Chem Soc (2018)

Asymmetric Palladium-Catalyzed Directed Intermolecular Fluoroarylation of Styrenes

由 Talbot, Eric P. A., Fernandes, Talita de A., McKenna, Jeffrey M., Toste, F. Dean
出版 2014

The development and mechanistic investigation of a palladium-catalyzed 1,3-arylfluorination of chromenes

由 Thornbury, Richard T., Saini, Vaneet, Fernandes, Talita de A., Santiago, Celine B., Talbot, Eric P. A., Sigman, Matthew S., McKenna, Jeffrey M., Toste, F. Dean
發表在 Chem Sci (2017)

Bardoxolone conjugation enables targeted protein degradation of BRD4

由 Tong, Bingqi, Luo, Mai, Xie, Yi, Spradlin, Jessica N., Tallarico, John A., McKenna, Jeffrey M., Schirle, Markus, Maimone, Thomas J., Nomura, Daniel K.
發表在 Sci Rep (2020)

Chemoproteomics-Enabled Discovery of Covalent RNF114-Based Degraders that Mimic Natural Product Function

由 Luo, Mai, Spradlin, Jessica N., Boike, Lydia, Tong, Bingqi, Brittain, Scott M., McKenna, Jeffrey M., Tallarico, John A., Schirle, Markus, Maimone, Thomas J., Nomura, Daniel K.
發表在 Cell Chem Biol (2021)

Discovery of a Functional Covalent Ligand Targeting an Intrinsically Disordered Cysteine Within MYC

由 Boike, Lydia, Cioffi, Alexander G., Majewski, Felix C., Co, Jennifer, Henning, Nathaniel J., Jones, Michael D., Liu, Gang, McKenna, Jeffrey M., Tallarico, John A., Schirle, Markus, Nomura, Daniel K.
發表在 Cell Chem Biol (2020)

Covalent Ligand Screening Uncovers a RNF4 E3 Ligase Recruiter for Targeted Protein Degradation Applications

由 Ward, Carl C., Kleinman, Jordan I., Brittain, Scott M., Lee, Patrick S., Sham Chung, Clive Yik, Kim, Kenneth, Petri, Yana, Thomas, Jason R., Tallarico, John A., McKenna, Jeffrey M., Schirle, Markus, Nomura, Daniel K.
發表在 ACS Chem Biol (2019)

Manumycin Polyketides Act as Molecular Glues Between UBR7 and P53

由 Isobe, Yosuke, Okumura, Mikiko, McGregor, Lynn M., Brittain, Scott M., Jones, Michael D., Liang, Xiaoyou, White, Ross, Forrester, William, McKenna, Jeffrey M., Tallarico, John A., Schirle, Markus, Maimone, Thomas J., Nomura, Daniel K.
發表在 Nat Chem Biol (2020)

A Nimbolide-Based Kinase Degrader Preferentially Degrades Oncogenic BCR-ABL

由 Tong, Bingqi, Spradlin, Jessica N., Novaes, Luiz F.T., Zhang, Erika, Hu, Xirui, Moeller, Malte, Brittain, Scott M., McGregor, Lynn M., McKenna, Jeffrey M., Tallarico, John A., Schirle, Markus, Maimone, Thomas J., Nomura, Daniel K.
發表在 ACS Chem Biol (2020)

Harnessing the Anti-Cancer Natural Product Nimbolide for Targeted Protein Degradation

由 Spradlin, Jessica N., Hu, Xirui, Ward, Carl C., Brittain, Scott M., Jones, Michael D., Ou, Lisha, To, Milton, Proudfoot, Andrew, Ornelas, Elizabeth, Woldegiorgis, Mikias, Olzmann, James A., Bussiere, Dirksen E., Thomas, Jason R., Tallarico, John A., McKenna, Jeffrey M., Schirle, Markus, Maimone, Thomas J., Nomura, Daniel K.
發表在 Nat Chem Biol (2019)