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Chemoproteomics-Enabled Discovery of Covalent RNF114-Based Degraders that Mimic Natural Product Function

The translation of functionally active natural products into fully synthetic small molecule mimetics has remained an important process in medicinal chemistry. We recently discovered that the terpene natural product nimbolide can be utilized as a covalent recruiter of the E3 ubiquitin ligase RNF114 f...

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Bibliografiske detaljer
Udgivet i:Cell Chem Biol
Main Authors: Luo, Mai, Spradlin, Jessica N., Boike, Lydia, Tong, Bingqi, Brittain, Scott M., McKenna, Jeffrey M., Tallarico, John A., Schirle, Markus, Maimone, Thomas J., Nomura, Daniel K.
Format: Artigo
Sprog:Inglês
Udgivet: 2021
Fag:
Online adgang:https://ncbi.nlm.nih.gov/pmc/articles/PMC8052289/
https://ncbi.nlm.nih.gov/pubmed/33513350
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.chembiol.2021.01.005
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