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Chemoproteomics-Enabled Covalent Ligand Screening Reveals a Thioredoxin-Caspase 3 Interaction Disruptor That Impairs Breast Cancer Pathogenicity

Covalent ligand discovery is a promising strategy to develop small-molecule effectors against therapeutic targets. Recent studies have shown that dichlorotriazines are promising reactive scaffolds that preferentially react with lysines. Here, we have synthesized a series of dichlorotriazine-based co...

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Pubblicato in:ACS Chem Biol
Autori principali: Anderson, Kimberly E., To, Milton, Olzmann, James A., Nomura, Daniel K.
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2017
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC6205226/
https://ncbi.nlm.nih.gov/pubmed/28892616
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acschembio.7b00711
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