Preparation of the Metabotropic Glutamate Receptor 5 (mGluR5) PET Tracer [(18)F]FPEB for Human Use: An Automated Radiosynthesis and a Novel One-Pot Synthesis of its Radiolabeling P...

Por Lim, Keunpoong, Labaree, David, Li, Songye, Huang, Yiyun
Publicado no Appl Radiat Isot (2014)

Synthesis and evaluation of 11β-(4-Substituted phenyl) estradiol analogs: Transition from estrogen receptor agonists to antagonists

Por Hanson, Robert N., Hua, Edward, Hendricks, J. Adam, Labaree, David, Hochberg, Richard B.
Publicado em 2012

Synthesis and Evaluation of 4-(Substituted styryl/alkenyl) -3,5-Bis(4-hydroxyphenyl)-isoxazoles as Ligands for the Estrogen Receptor

Por Haddad, Terra, Gershman, Rachel, Dilis, Robert, Labaree, David, Hochberg, Richard B., Hanson, Robert N.
Publicado em 2012

Synthesis and Evaluation of 17α-(Dimethylphenyl)vinyl Estradiols as Probes of the Estrogen Receptor-α Ligand Binding Domain

Por Hanson, Robert N., McCaskill, Emmett, Tongcharoensirikul, Pakamas, Dilis, Robert, Labaree, David, Hochberg, Richard B.
Publicado em 2012

Development and In Vivo Evaluation of a κ-Opioid Receptor Agonist as a PET Radiotracer with Superior Imaging Characteristics

Por Li, Songye, Zheng, Ming-Qiang, Naganawa, Mika, Kim, Sujin, Gao, Hong, Kapinos, Michael, Labaree, David, Huang, Yiyun
Publicado no J Nucl Med (2019)

Synthesis and evaluation of 17α-E-20-(heteroaryl)norpregn-1,3,5(10),20 tetraene-3,17β-diols [17α- (heteroaryl)vinyl estradiols] as ligands for the estrogen receptor-α-ligand bindin...

Por Olmsted, Sandra L., Tongcharoensirikul, Pakamas, McCaskill, Emmett, Gandiaga, Karla, Labaree, David, Hochberg, Richard B., Hanson, Robert N.
Publicado em 2011

Convergent synthesis of a steroidal antiestrogen-mitomycin C hybrid using “click” chemistry()

Por Hanson, Robert N., Hua, Edward, Labaree, David, Hochberg, Richard B., Proffitt, Kyle, Essigmann, John M., Croy, Robert G.
Publicado em 2012

Studies of the Metabotropic Glutamate Receptor 5 Radioligand [(11)C]ABP688 with N-acetylcysteine Challenge in Rhesus Monkeys

Por Sandiego, Christine M., Nabulsi, Nabeel, Lin, Shu-fei, Labaree, David, Najafzadeh, Soheila, Huang, Yiyun, Cosgrove, Kelly, Carson, Richard E.
Publicado em 2013

Binge alcohol use is not associated with alterations in striatal dopamine receptor binding or dopamine release

Por Wai, Jonathan M., Grassetti, Alexander, Slifstein, Mark, Matuskey, David, Nabulsi, Nabeel, Ropchan, Jim, Labaree, David, Huang, Yiyun, Martinez, Diana
Publicado no Drug Alcohol Depend (2019)

Targeting the Estrogen Receptor with Metal-carbonyl Derivatives of Estradiol

Por Hanson, Robert N., Kirss, Rein, McCaskill, Emmett, Hua, Edward, Tongcharoensirikul, Pakamas, Olmsted, Sandra L., Labaree, David, Hochberg, Richard B.
Publicado em 2012

Kinetic analysis of drug–target interactions with PET for characterization of pharmacological hysteresis

Por Salinas, Cristian, Weinzimmer, David, Searle, Graham, Labaree, David, Ropchan, Jim, Huang, Yiyun, Rabiner, Eugenii A, Carson, Richard E, Gunn, Roger N
Publicado em 2013

Determination of the In vivo Selectivity of a new Kappa Opioid Receptor Antagonist PET Tracer [(11)C]LY2795050 in the Rhesus Monkey

Por Kim, Su Jin, Zheng, Ming-Qiang, Nabulsi, Nabeel, Labaree, David, Ropchan, Jim, Najafzadeh, Soheila, Carson, Richard E., Huang, Yiyun, Morris, Evan D.
Publicado no J Nucl Med (2013)

Separating dopamine D(2) and D(3) receptor sources of [(11)C]-(+)-PHNO binding potential: independent component analysis of competitive binding

Por Smart, Kelly, Gallezot, Jean-Dominique, Nabulsi, Nabeel, Labaree, David, Zheng, Ming-Qiang, Huang, Yiyun, Carson, Richard E., Hillmer, Ansel T., Worhunsky, Patrick D.
Publicado no Neuroimage (2020)

Evaluation of pancreatic VMAT2 binding with active and inactive enantiomers of (18)F-FP-DTBZ in baboons

Por Naganawa, Mika, Lin, Shu-fei, Lim, Keunpoong, Labaree, David, Ropchan, Jim, Harris, Paul, Huang, Yiyun, Ichise, Masanori, Carson, Richard E., Cline, Gary W.
Publicado no Nucl Med Biol (2016)

Synthesis and in Vivo Evaluation of a Novel PET Radiotracer for Imaging of Synaptic Vesicle Glycoprotein 2A (SV2A) in Nonhuman Primates

Por Li, Songye, Cai, Zhengxin, Wu, Xiaoai, Holden, Daniel, Pracitto, Richard, Kapinos, Michael, Gao, Hong, Labaree, David, Nabulsi, Nabeel, Carson, Richard E., Huang, Yiyun
Publicado no ACS Chem Neurosci (2018)

Binding of the synaptic vesicle radiotracer [(11)C]UCB-J is unchanged during functional brain activation using a visual stimulation task

Por Smart, Kelly, Liu, Heather, Matuskey, David, Chen, Ming-Kai, Torres, Kristen, Nabulsi, Nabeel, Labaree, David, Ropchan, Jim, Hillmer, Ansel T, Huang, Yiyun, Carson, Richard E
Publicado no J Cereb Blood Flow Metab (2020)

PARAMETRIC IMAGING AND TEST-RETEST VARIABILITY OF (11)C-(+)-PHNO BINDING TO D(2)/D(3) DOPAMINE RECEPTORS IN HUMANS ON THE HRRT PET SCANNER

Por Gallezot, Jean-Dominique, Zheng, Ming-Qiang, Lim, Keunpoong, Lin, Shu-fei, Labaree, David, Matuskey, David, Huang, Yiyun, Ding, Yu-Shin, Carson, Richard E., Malison, Robert T.
Publicado em 2014

Sex Differences in the Brain's Dopamine Signature of Cigarette Smoking

Por Cosgrove, Kelly P., Wang, Shuo, Kim, Su-Jin, McGovern, Erin, Nabulsi, Nabeel, Gao, Hong, Labaree, David, Tagare, Hemant D., Sullivan, Jenna M., Morris, Evan D.
Publicado no J Neurosci (2014)

PET Imaging of the Effects of Age and Cocaine on the Norepinephrine Transporter in the Human Brain Using (S,S)-[(11)C]O-Methylreboxetine and HRRT

Por Ding, Yu-Shin, Singhal, Tarun, Planeta-Wilson, Beata, Gallezot, Jean-Dominique, Nabulsi, Nabeel, Labaree, David, Ropchan, Jim, Henry, Shannan, Williams, Wendol, Carson, Richard, Neumeister, Alexander, Malison, Robert T.
Publicado em 2010

Tracer kinetic modeling of [(11)C]AFM, a new PET imaging agent for the serotonin transporter

Por Naganawa, Mika, Nabulsi, Nabeel, Planeta, Beata, Gallezot, Jean-Dominique, Lin, Shu-Fei, Najafzadeh, Soheila, Williams, Wendol, Ropchan, Jim, Labaree, David, Neumeister, Alexander, Huang, Yiyun, Carson, Richard E
Publicado em 2013