Preparation of the Metabotropic Glutamate Receptor 5 (mGluR5) PET Tracer [(18)F]FPEB for Human Use: An Automated Radiosynthesis and a Novel One-Pot Synthesis of its Radiolabeling P...

par Lim, Keunpoong, Labaree, David, Li, Songye, Huang, Yiyun
Publié dans Appl Radiat Isot (2014)

Synthesis and evaluation of 11β-(4-Substituted phenyl) estradiol analogs: Transition from estrogen receptor agonists to antagonists

par Hanson, Robert N., Hua, Edward, Hendricks, J. Adam, Labaree, David, Hochberg, Richard B.
Publié 2012

Synthesis and Evaluation of 4-(Substituted styryl/alkenyl) -3,5-Bis(4-hydroxyphenyl)-isoxazoles as Ligands for the Estrogen Receptor

par Haddad, Terra, Gershman, Rachel, Dilis, Robert, Labaree, David, Hochberg, Richard B., Hanson, Robert N.
Publié 2012

Synthesis and Evaluation of 17α-(Dimethylphenyl)vinyl Estradiols as Probes of the Estrogen Receptor-α Ligand Binding Domain

par Hanson, Robert N., McCaskill, Emmett, Tongcharoensirikul, Pakamas, Dilis, Robert, Labaree, David, Hochberg, Richard B.
Publié 2012

Development and In Vivo Evaluation of a κ-Opioid Receptor Agonist as a PET Radiotracer with Superior Imaging Characteristics

par Li, Songye, Zheng, Ming-Qiang, Naganawa, Mika, Kim, Sujin, Gao, Hong, Kapinos, Michael, Labaree, David, Huang, Yiyun
Publié dans J Nucl Med (2019)

Synthesis and evaluation of 17α-E-20-(heteroaryl)norpregn-1,3,5(10),20 tetraene-3,17β-diols [17α- (heteroaryl)vinyl estradiols] as ligands for the estrogen receptor-α-ligand bindin...

par Olmsted, Sandra L., Tongcharoensirikul, Pakamas, McCaskill, Emmett, Gandiaga, Karla, Labaree, David, Hochberg, Richard B., Hanson, Robert N.
Publié 2011

Convergent synthesis of a steroidal antiestrogen-mitomycin C hybrid using “click” chemistry()

par Hanson, Robert N., Hua, Edward, Labaree, David, Hochberg, Richard B., Proffitt, Kyle, Essigmann, John M., Croy, Robert G.
Publié 2012

Studies of the Metabotropic Glutamate Receptor 5 Radioligand [(11)C]ABP688 with N-acetylcysteine Challenge in Rhesus Monkeys

par Sandiego, Christine M., Nabulsi, Nabeel, Lin, Shu-fei, Labaree, David, Najafzadeh, Soheila, Huang, Yiyun, Cosgrove, Kelly, Carson, Richard E.
Publié 2013

Binge alcohol use is not associated with alterations in striatal dopamine receptor binding or dopamine release

par Wai, Jonathan M., Grassetti, Alexander, Slifstein, Mark, Matuskey, David, Nabulsi, Nabeel, Ropchan, Jim, Labaree, David, Huang, Yiyun, Martinez, Diana
Publié dans Drug Alcohol Depend (2019)

Targeting the Estrogen Receptor with Metal-carbonyl Derivatives of Estradiol

par Hanson, Robert N., Kirss, Rein, McCaskill, Emmett, Hua, Edward, Tongcharoensirikul, Pakamas, Olmsted, Sandra L., Labaree, David, Hochberg, Richard B.
Publié 2012

Kinetic analysis of drug–target interactions with PET for characterization of pharmacological hysteresis

par Salinas, Cristian, Weinzimmer, David, Searle, Graham, Labaree, David, Ropchan, Jim, Huang, Yiyun, Rabiner, Eugenii A, Carson, Richard E, Gunn, Roger N
Publié 2013

Determination of the In vivo Selectivity of a new Kappa Opioid Receptor Antagonist PET Tracer [(11)C]LY2795050 in the Rhesus Monkey

par Kim, Su Jin, Zheng, Ming-Qiang, Nabulsi, Nabeel, Labaree, David, Ropchan, Jim, Najafzadeh, Soheila, Carson, Richard E., Huang, Yiyun, Morris, Evan D.
Publié dans J Nucl Med (2013)

Separating dopamine D(2) and D(3) receptor sources of [(11)C]-(+)-PHNO binding potential: independent component analysis of competitive binding

par Smart, Kelly, Gallezot, Jean-Dominique, Nabulsi, Nabeel, Labaree, David, Zheng, Ming-Qiang, Huang, Yiyun, Carson, Richard E., Hillmer, Ansel T., Worhunsky, Patrick D.
Publié dans Neuroimage (2020)

Evaluation of pancreatic VMAT2 binding with active and inactive enantiomers of (18)F-FP-DTBZ in baboons

par Naganawa, Mika, Lin, Shu-fei, Lim, Keunpoong, Labaree, David, Ropchan, Jim, Harris, Paul, Huang, Yiyun, Ichise, Masanori, Carson, Richard E., Cline, Gary W.
Publié dans Nucl Med Biol (2016)

Synthesis and in Vivo Evaluation of a Novel PET Radiotracer for Imaging of Synaptic Vesicle Glycoprotein 2A (SV2A) in Nonhuman Primates

par Li, Songye, Cai, Zhengxin, Wu, Xiaoai, Holden, Daniel, Pracitto, Richard, Kapinos, Michael, Gao, Hong, Labaree, David, Nabulsi, Nabeel, Carson, Richard E., Huang, Yiyun
Publié dans ACS Chem Neurosci (2018)

Binding of the synaptic vesicle radiotracer [(11)C]UCB-J is unchanged during functional brain activation using a visual stimulation task

par Smart, Kelly, Liu, Heather, Matuskey, David, Chen, Ming-Kai, Torres, Kristen, Nabulsi, Nabeel, Labaree, David, Ropchan, Jim, Hillmer, Ansel T, Huang, Yiyun, Carson, Richard E
Publié dans J Cereb Blood Flow Metab (2020)

PARAMETRIC IMAGING AND TEST-RETEST VARIABILITY OF (11)C-(+)-PHNO BINDING TO D(2)/D(3) DOPAMINE RECEPTORS IN HUMANS ON THE HRRT PET SCANNER

par Gallezot, Jean-Dominique, Zheng, Ming-Qiang, Lim, Keunpoong, Lin, Shu-fei, Labaree, David, Matuskey, David, Huang, Yiyun, Ding, Yu-Shin, Carson, Richard E., Malison, Robert T.
Publié 2014

Sex Differences in the Brain's Dopamine Signature of Cigarette Smoking

par Cosgrove, Kelly P., Wang, Shuo, Kim, Su-Jin, McGovern, Erin, Nabulsi, Nabeel, Gao, Hong, Labaree, David, Tagare, Hemant D., Sullivan, Jenna M., Morris, Evan D.
Publié dans J Neurosci (2014)

PET Imaging of the Effects of Age and Cocaine on the Norepinephrine Transporter in the Human Brain Using (S,S)-[(11)C]O-Methylreboxetine and HRRT

par Ding, Yu-Shin, Singhal, Tarun, Planeta-Wilson, Beata, Gallezot, Jean-Dominique, Nabulsi, Nabeel, Labaree, David, Ropchan, Jim, Henry, Shannan, Williams, Wendol, Carson, Richard, Neumeister, Alexander, Malison, Robert T.
Publié 2010

Tracer kinetic modeling of [(11)C]AFM, a new PET imaging agent for the serotonin transporter

par Naganawa, Mika, Nabulsi, Nabeel, Planeta, Beata, Gallezot, Jean-Dominique, Lin, Shu-Fei, Najafzadeh, Soheila, Williams, Wendol, Ropchan, Jim, Labaree, David, Neumeister, Alexander, Huang, Yiyun, Carson, Richard E
Publié 2013