Chiral resolution and absolute configuration of the enantiomers of the psychoactive “designer drug” 3,4-methylenedioxypyrovalerone

Por Suzuki, Masaki, Deschamps, Jeffrey R., Jacobson, Arthur E., Rice, Kenner C.
Publicado no Chirality (2015)

PROBES FOR NARCOTIC RECEPTOR MEDIATED PHENOMENA. 38.(1) AN EXPEDITIOUS SYNTHESIS OF RAC-CIS-4a-ETHYL-2-METHYL-1,2,3,4,4a,9a-HEXAHYDROBENZOFURO[2,3-c]PYRIDIN-6-OL AND RAC-CIS-2-METH...

Por Iyer, Malliga R., Deschamps, Jeffrey R., Jacobson, Arthur E., Rice, Kenner C.
Publicado em 2009

Diastereoselective One-Pot Synthesis of 7- and 8-Substituted 5-Phenylmorphans

Por Lim, Hwan Jung, Deschamps, Jeffrey R., Jacobson, Arthur E., Rice, Kenner C.
Publicado em 2011

Synthesis of Enantiopure 10-Nornaltrexones in the Search for Toll-like Receptor 4 Antagonists and Opioid Ligands

Por Selfridge, Brandon R., Deschamps, Jeffrey R., Jacobson, Arthur E., Rice, Kenner C.
Publicado em 2014

Z and E rotamers of N-formyl-1-bromo-4-hydroxy-3-methoxymorphinan-6-one and their interconversion as studied by (1)H/(13)C NMR spectroscopy and quantum chemical calculations

Por Sulima, Agnieszka, Cheng, Kejun, Jacobson, Arthur E., Rice, Kenner C., Gawrisch, Klaus, Lee, Yong-Sok
Publicado em 2012

Probes for narcotic receptor mediated phenomena. 47.(1) Novel C4a- and N-substituted-1,2,3,4,4a,9a-hexahydrobenzofuro[2,3-c] pyridin-6-ols

Por Iyer, Malliga R., Rothman, Richard B., Dersch, Christina M., Jacobson, Arthur E., Rice, Kenner C.
Publicado em 2013

Probes for narcotic receptor mediated phenomena 49. N-Substituted rac-cis-4a-arylalkyl-1,2,3,4,4a,9a-hexahydrobenzofuro[2,3-c]pyridin-6-ols

Por Iyer, Malliga R., Rothman, Richard B., Dersch, Christina M., Jacobson, Arthur E., Rice, Kenner C.
Publicado no Eur J Med Chem (2015)

Configurational Reassignment and Improved Preparation of the Competitive IL-6 Receptor Antagonist 20R,21R-Epoxyresibufogenin-3-formate

Por Boos, Terrence L., Cheng, Kejun, Greiner, Elisabeth, Deschamps, Jeffrey R., Jacobson, Arthur E., Rice, Kenner C.
Publicado em 2012

Synthesis of 2-(5Z,8Z,11Z,14Z)-Icosa-5,8,11,14-tetraenamidoethyl-d(4) Dihydrogen Phosphate, Tetra-deuterated pAEA

Por Cheng, Kejun, Saha, Bijali, Mahadevan, A., Razdan, Raj K., Kunos, George, Jacobson, Arthur E., Rice, Kenner C.
Publicado em 2008

Evidence for Non-Competitive Modulation of Substrate-Induced Serotonin Release

Por Rothman, Richard B., Baumann, Michael H., Blough, Bruce E., Jacobson, Arthur E., Rice, Kenner C., Partilla, John S.
Publicado em 2010

Probes for narcotic receptor mediated phenomena. 48. C7- and C8-Substituted 5-phenylmorphan opioids from diastereoselective alkylation

Por Lim, Hwan Jung, Dersch, Christina M., Rothman, Richard B., Deschamps, Jeffrey R., Jacobson, Arthur E., Rice, Kenner C.
Publicado em 2013

Design and Synthesis of 2- and 3-Substituted-3-phenylpropyl Analogs of 1-[2-[Bis(4-fluorophenyl)methoxy]ethyl]-4-(3-phenylpropyl)piperazine and 1-[2-(Diphenylmethoxy)ethyl]-4-(3-ph...

Por Hsin, Ling-Wei, Chang, Li-Te, Rothman, Richard B., Dersch, Christina M., Jacobson, Arthur E., Rice, Kenner C.
Publicado no J Med Chem (2008)

Probes for Narcotic Receptor Mediated Phenomena. 39.1 Enantiomeric N-Substituted Benzofuro[2,3-c]pyridin-6-ols: Synthesis and Topological Relationship to Oxide-bridged Phenylmorpha...

Por Zhang, Yi, Lee, Yong Sok, Rothman, Richard B., Dersch, Christina M., Deschamps, Jeffrey R., Jacobson, Arthur E., Rice, Kenner C.
Publicado em 2009

Probes for narcotic receptor mediated phenomena. 41. Unusual inverse μ-agonists and potent μ-opioid antagonists by modification of the N-substituent in enantiomeric 5-(3- hydroxyph...

Por Cheng, Kejun, Lee, Yong Sok, Rothman, Richard B., Dersch, Christina M., Bittman, Ross W., Jacobson, Arthur E., Rice, Kenner C.
Publicado em 2011

Probes for narcotic receptor mediated phenomena. 46. N-Substituted-2,3,4,9,10,10a-hexahydro-1H-1,4a-(epiminoethano)phenanthren-6- and 8-ols - carbocyclic relatives of f-oxide bridg...

Por Li, Fuying, Deck, Jason A., Dersch, Christina M., Rothman, Richard B., Deschamps, Jeffrey R., Jacobson, Arthur E., Rice, Kenner C.
Publicado em 2012

Probes for narcotic receptor mediated phenomena. 40.(1 )N-Substituted cis-4a-ethyl-1,2,3,4,4a,9a-hexahydrobenzofuro[2,3-c]pyridin-8-ols

Por Iyer, Malliga R., Lee, Yong Sok, Deschamps, Jeffrey R., Rothman, Richard B., Dersch, Christina M., Jacobson, Arthur E., Rice, Kenner C.
Publicado em 2009

Probes for narcotic receptor mediated phenomena. 44. Synthesis of an N-substituted 4-hydroxy-5-(3-hydroxyphenyl)morphan with high affinity and selective μ-antagonist activity

Por Iyer, Malliga R., Lee, Yong Sok, Deschamps, Jeffrey R., Dersch, Christina M., Rothman, Richard B., Jacobson, Arthur E., Rice, Kenner C.
Publicado em 2012

Structure-Activity Relationships of (+)-Naltrexone-Inspired Toll-Like Receptor 4 (TLR4) Antagonists

Por Selfridge, Brandon R., Wang, Xiaohui, Zhang, Yingning, Yin, Hang, Grace, Peter M., Watkins, Linda R., Jacobson, Arthur E., Rice, Kenner C.
Publicado no J Med Chem (2015)

Probes for narcotic receptor mediated phenomena. 42. Synthesis and in vitro pharmacological characterization of the N-methyl and N-phenethyl analogues of the racemic ortho-c and pa...

Por Kim, Jin-Hee, Deschamps, Jeffrey R., Rothman, Richard B., Dersch, Christina M., Folk, John E., Cheng, Kejun, Jacobson, Arthur E., Rice, Kenner C.
Publicado em 2011

A simple nonradioactive method for the determination of the binding affinities of antibodies induced by hapten bioconjugates for drugs of abuse

Por Torres, Oscar B., Antoline, Joshua F. G., Li, Fuying, Jalah, Rashmi, Jacobson, Arthur E., Rice, Kenner C., Alving, Carl R., Matyas, Gary R.
Publicado no Anal Bioanal Chem (2015)