Considerations for improved performance of competition association assays analysed with the Motulsky–Mahan's “kinetics of competitive binding” model

Por Georgi, Victoria, Dubrovskiy, Alexey, Steigele, Stephan, Fernández‐Montalván, Amaury E.
Publicado no Br J Pharmacol (2019)

Characterization of 12 GnRH peptide agonists – a kinetic perspective

Por Nederpelt, Indira, Georgi, Victoria, Schiele, Felix, Nowak‐Reppel, Katrin, Fernández‐Montalván, Amaury E., IJzerman, Adriaan P., Heitman, Laura H.
Publicado no Br J Pharmacol (2015)

Halogen–Aromatic π Interactions Modulate Inhibitor Residence Times

Por Heroven, Christina, Georgi, Victoria, Ganotra, Gaurav K., Brennan, Paul, Wolfreys, Finn, Wade, Rebecca C., Fernández-Montalván, Amaury E., Chaikuad, Apirat, Knapp, Stefan
Publicado no Angew Chem Int Ed Engl (2018)

Probe dependency in the determination of ligand binding kinetics at a prototypical G protein-coupled receptor

Por Bosma, Reggie, Stoddart, Leigh A., Georgi, Victoria, Bouzo-Lorenzo, Monica, Bushby, Nick, Inkoom, Loretta, Waring, Michael J., Briddon, Stephen J., Vischer, Henry F., Sheppard, Robert J., Fernández-Montalván, Amaury, Hill, Stephen J., Leurs, Rob
Publicado no Sci Rep (2019)

In vitro and in silico analysis of the effects of D (2) receptor antagonist target binding kinetics on the cellular response to fluctuating dopamine concentrations

Por de Witte, Wilhelmus E A, Versfelt, Joost W, Kuzikov, Maria, Rolland, Solene, Georgi, Victoria, Gribbon, Philip, Gul, Sheraz, Huntjens, Dymphy, van der Graaf, Piet Hein, Danhof, Meindert, Fernández‐Montalván, Amaury, Witt, Gesa, de Lange, Elizabeth C M
Publicado no Br J Pharmacol (2018)