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Structure-Activity Relationships of Pyrimidine Nucleotides Containing a 5′-α,β-Methylene Diphosphonate at the P2Y(6) Receptor

The G(q)-coupled P2Y(6) receptor (P2Y(6)R) is a component of the purinergic signaling system and functions in inflammatory, cardiovascular and metabolic processes. UDP, the native P2Y(6)R agonist and P2Y(14)R partial agonist, is subject to hydrolysis by ectonucleotidases. Therefore, we have synthesi...

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Bibliografiske detaljer
Udgivet i:Bioorg Med Chem Lett
Main Authors: Oliva, Paola, Scortichini, Mirko, Dobelmann, Clemens, Jain, Shanu, Gopinatth, Varun, Toti, Kiran S., Phung, Ngan B., Junker, Anna, Jacobson, Kenneth A.
Format: Artigo
Sprog:Inglês
Udgivet: 2021
Fag:
Online adgang:https://ncbi.nlm.nih.gov/pmc/articles/PMC8276771/
https://ncbi.nlm.nih.gov/pubmed/34048882
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmcl.2021.128137
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