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Structure Activity Relationship of 3-Nitro-2-(trifluoromethyl)-2H-chromene Derivatives as P2Y(6) Receptor Antagonists

Various 6-alkynyl analogues of a known 3-nitro-2-(trifluoromethyl)-2H-chromene antagonist 3 of the G(q)-coupled P2Y(6) receptor (P2Y(6)R) were synthesized using a Sonogashira reaction to replace a 6-iodo group. The analogues were tested in a functional assay consisting of inhibition of calcium mobil...

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Detalhes bibliográficos
Publicado no:Bioorg Med Chem Lett
Main Authors: Jung, Young-Hwan, Jain, Shanu, Gopinatth, Varun, Phung, Ngan B., Gao, Zhan-Guo, Jacobson, Kenneth A.
Formato: Artigo
Idioma:Inglês
Publicado em: 2021
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC8240625/
https://ncbi.nlm.nih.gov/pubmed/33831560
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmcl.2021.128008
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