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Structure-Activity Relationships of Pyrimidine Nucleotides Containing a 5′-α,β-Methylene Diphosphonate at the P2Y(6) Receptor

The G(q)-coupled P2Y(6) receptor (P2Y(6)R) is a component of the purinergic signaling system and functions in inflammatory, cardiovascular and metabolic processes. UDP, the native P2Y(6)R agonist and P2Y(14)R partial agonist, is subject to hydrolysis by ectonucleotidases. Therefore, we have synthesi...

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Bibliografski detalji
Izdano u:Bioorg Med Chem Lett
Glavni autori: Oliva, Paola, Scortichini, Mirko, Dobelmann, Clemens, Jain, Shanu, Gopinatth, Varun, Toti, Kiran S., Phung, Ngan B., Junker, Anna, Jacobson, Kenneth A.
Format: Artigo
Jezik:Inglês
Izdano: 2021
Teme:
Online pristup:https://ncbi.nlm.nih.gov/pmc/articles/PMC8276771/
https://ncbi.nlm.nih.gov/pubmed/34048882
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmcl.2021.128137
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