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Selective Photoswitchable Allosteric Agonist of a G Protein-Coupled Receptor

[Image: see text] G protein-coupled receptors (GPCRs) are the most common targets of drug discovery. However, the similarity between related GPCRs combined with the complex spatiotemporal dynamics of receptor activation in vivo has hindered drug development. Photopharmacology offers the possibility...

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Détails bibliographiques
Publié dans:J Am Chem Soc
Auteurs principaux: Donthamsetti, Prashant, Konrad, David B., Hetzler, Belinda, Fu, Zhu, Trauner, Dirk, Isacoff, Ehud Y.
Format: Artigo
Langue:Inglês
Publié: American Chemical Society 2021
Accès en ligne:https://ncbi.nlm.nih.gov/pmc/articles/PMC8227462/
https://ncbi.nlm.nih.gov/pubmed/34115935
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/jacs.1c02586
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