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Proteolysis targeting chimeras (PROTACs) come of age: entering the third decade of targeted protein degradation

With the discovery of PROteolysis TArgeting Chimeras (PROTACs) twenty years ago, targeted protein degradation (TPD) has changed the landscape of drug development. PROTACs have evolved from cell-impermeable peptide-small molecule chimeras to orally bioavailable clinical candidate drugs that degrade o...

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Wedi'i Gadw mewn:
Manylion Llyfryddiaeth
Cyhoeddwyd yn:RSC Chem Biol
Prif Awduron: Bond, Michael J., Crews, Craig M.
Fformat: Artigo
Iaith:Inglês
Cyhoeddwyd: RSC 2021
Pynciau:
Mynediad Ar-lein:https://ncbi.nlm.nih.gov/pmc/articles/PMC8190915/
https://ncbi.nlm.nih.gov/pubmed/34212149
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1039/d1cb00011j
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