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Mechanism of gating and partial agonist action in the glycine receptor

Ligand-gated ion channels mediate signal transduction at chemical synapses and transition between resting, open and desensitized states in response to neurotransmitter binding. Neurotransmitters that produce maximum open channel probabilities (Po) are full agonists whereas those that yield lower tha...

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Publicat a:Cell
Autors principals: Yu, Jie, Zhu, Hongtao, Lape, Remigijus, Greiner, Timo, Du, Juan, Lü, Wei, Sivilotti, Lucia, Gouaux, Eric
Format: Artigo
Idioma:Inglês
Publicat: 2021
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC8115384/
https://ncbi.nlm.nih.gov/pubmed/33567265
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.cell.2021.01.026
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