Cargando...

Therapeutic Opportunities of Targeting Allosteric Binding Sites on the Calcium-Sensing Receptor

[Image: see text] The CaSR is a class C G protein-coupled receptor (GPCR) that acts as a multimodal chemosensor to maintain diverse homeostatic functions. The CaSR is a clinical therapeutic target in hyperparathyroidism and has emerged as a putative target in several other diseases. These include hy...

Descripción completa

Guardado en:
Detalles Bibliográficos
Publicado en:ACS Pharmacol Transl Sci
Autores principales: Diao, Jiayin, DeBono, Aaron, Josephs, Tracy M., Bourke, Jane E., Capuano, Ben, Gregory, Karen J., Leach, Katie
Formato: Artigo
Lenguaje:Inglês
Publicado: American Chemical Society 2021
Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC8033781/
https://ncbi.nlm.nih.gov/pubmed/33860192
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acsptsci.1c00046
Etiquetas: Agregar Etiqueta
Sin Etiquetas, Sea el primero en etiquetar este registro!