Lataa...
4-Benzylideneisoquinoline-1,3(2H,4H)-diones as tyrosyl DNA phosphodiesterase 2 (TDP2) inhibitors
Tyrosyl-DNA phosphodiesterase 2 (TDP2) repairs topoisomerase II (Top2) mediated DNA damages, including double-strand breaks (DSBs) that underpin the anticancer mechanism of clinical TOP2 poisons such as etoposide (ETP). Inhibition of TDP2 could sensitize cancer cells toward TOP2 poisons by increasin...
Tallennettuna:
| Julkaisussa: | Med Chem Res |
|---|---|
| Päätekijät: | , , , , |
| Aineistotyyppi: | Artigo |
| Kieli: | Inglês |
| Julkaistu: |
2020
|
| Aiheet: | |
| Linkit: | https://ncbi.nlm.nih.gov/pmc/articles/PMC7993140/ https://ncbi.nlm.nih.gov/pubmed/33776385 https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1007/s00044-020-02662-w |
| Tagit: |
Lisää tagi
Ei tageja, Lisää ensimmäinen tagi!
|