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Novel Deazaflavin Tyrosyl-DNA Phosphodiesterase 2 (TDP2) Inhibitors

Tyrosyl-DNA phosphodiesterase 2 (TDP2) is a DNA repair enzyme that removes 5′-phosphotyrosyl blockages resulting from topoisomerase II (TOP2)-DNA cleavage complexes trapped by TOP2 inhibitors. TDP2 is a logical target for the development of therapeutics to complement existing treatments based on inh...

पूर्ण विवरण

में बचाया:
ग्रंथसूची विवरण
में प्रकाशित:DNA Repair (Amst)
मुख्य लेखकों: Kiselev, Evgeny, Ravji, Azhar, Kankanala, Jayakanth, Xie, Jiashu, Wang, Zhengqiang, Pommier, Yves
स्वरूप: Artigo
भाषा:Inglês
प्रकाशित: 2019
विषय:
ऑनलाइन पहुंच:https://ncbi.nlm.nih.gov/pmc/articles/PMC6952553/
https://ncbi.nlm.nih.gov/pubmed/31775111
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.dnarep.2019.102747
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