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Insights into Current Tropomyosin Receptor Kinase (TRK) Inhibitors: Development and Clinical Application

The use of kinase-directed precision medicine has been heavily pursued since the discovery and development of imatinib. Annually, it is estimated that around ~20 000 new cases of tropomyosin receptor kinase (TRK) cancers are diagnosed, with the majority of cases exhibiting a TRK genomic rearrangemen...

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Detalhes bibliográficos
Publicado no:J Med Chem
Main Authors: Yan, Wei, Lakkaniga, Naga Rajiv, Carlomagno, Francesca, Santoro, Massimo, McDonald, Neil Q., Lv, Fengping, Gunaganti, Naresh, Frett, Brendan, Li, Hong-yu
Formato: Artigo
Idioma:Inglês
Publicado em: 2018
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC7875308/
https://ncbi.nlm.nih.gov/pubmed/30188734
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.jmedchem.8b01092
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