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The role of specific ATP-binding cassette transporters in the acquired resistance to pyrrolobenzodiazepine dimer-containing antibody-drug conjugates

Antibody drug conjugates (ADCs) containing pyrrolobenzodiazepine (PBD) dimers are being evaluated clinically in both hematological and solid tumors. These include ADCT-301 (camidanlumab tesirine) and ADCT-402 (loncastuximab tesirine) in pivotal Phase 2 trials that contain the payload tesirine which...

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Bibliografiske detaljer
Udgivet i:Mol Cancer Ther
Main Authors: Corbett, Simon, Huang, Shiran, Zammarchi, Francesca, Howard, Philip W, van Berkel, Patrick H, Hartley, John A
Format: Artigo
Sprog:Inglês
Udgivet: 2020
Fag:
Online adgang:https://ncbi.nlm.nih.gov/pmc/articles/PMC7611352/
https://ncbi.nlm.nih.gov/pubmed/32669316
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1158/1535-7163.MCT-20-0222
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