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Effects of Multiple Doses of Dichloroacetate on GSTZ1 Expression and Activity in Liver and Extrahepatic Tissues of Young and Adult Rats

Glutathione transferase zeta 1 (GSTZ1), expressed in liver and several extrahepatic tissues, catalyzes dechlorination of dichloroacetate (DCA) to glyoxylate. DCA inactivates GSTZ1, leading to autoinhibition of its metabolism. DCA is an investigational drug for treating several congenital and acquire...

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Bibliographic Details
Published in:Drug Metab Dispos
Main Authors: Squirewell, Edwin J., Smeltz, Marci G., Rowland-Faux, Laura, Horne, Lloyd P., Stacpoole, Peter W., James, Margaret O.
Format: Artigo
Language:Inglês
Published: The American Society for Pharmacology and Experimental Therapeutics 2020
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Online Access:https://ncbi.nlm.nih.gov/pmc/articles/PMC7589944/
https://ncbi.nlm.nih.gov/pubmed/32873593
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/dmd.120.000142
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