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Effects of Multiple Doses of Dichloroacetate on GSTZ1 Expression and Activity in Liver and Extrahepatic Tissues of Young and Adult Rats

Glutathione transferase zeta 1 (GSTZ1), expressed in liver and several extrahepatic tissues, catalyzes dechlorination of dichloroacetate (DCA) to glyoxylate. DCA inactivates GSTZ1, leading to autoinhibition of its metabolism. DCA is an investigational drug for treating several congenital and acquire...

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Publicat a:Drug Metab Dispos
Autors principals: Squirewell, Edwin J., Smeltz, Marci G., Rowland-Faux, Laura, Horne, Lloyd P., Stacpoole, Peter W., James, Margaret O.
Format: Artigo
Idioma:Inglês
Publicat: The American Society for Pharmacology and Experimental Therapeutics 2020
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC7589944/
https://ncbi.nlm.nih.gov/pubmed/32873593
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/dmd.120.000142
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