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Caffeine inhibits Notum activity by binding at the catalytic pocket

Notum inhibits Wnt signalling via enzymatic delipidation of Wnt ligands. Restoration of Wnt signalling by small molecule inhibition of Notum may be of therapeutic benefit in a number of pathologies including Alzheimer’s disease. Here we report Notum activity can be inhibited by caffeine (IC(50) 19 µ...

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Publicat a:Commun Biol
Autors principals: Zhao, Yuguang, Ren, Jingshan, Hillier, James, Lu, Weixian, Jones, Edith Yvonne
Format: Artigo
Idioma:Inglês
Publicat: Nature Publishing Group UK 2020
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC7544826/
https://ncbi.nlm.nih.gov/pubmed/33033363
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/s42003-020-01286-5
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