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Design and in vivo activity of A(3) adenosine receptor agonist prodrugs

Prodrugs (MRS7422, MRS7476) of highly selective A(3) adenosine receptor (AR) agonists Cl-IB-MECA and MRS5698, respectively, were synthesized by succinylation of the 2′ and 3′ hydroxyl groups, and the parent, active drug was shown to be readily liberated upon incubation with liver esterases. The prod...

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Detalhes bibliográficos
Publicado no:Purinergic Signal
Main Authors: Suresh, R. Rama, Jain, Shanu, Chen, Zhoumou, Tosh, Dilip K., Ma, Yanling, Podszun, Maren C., Rotman, Yaron, Salvemini, Daniela, Jacobson, Kenneth A.
Formato: Artigo
Idioma:Inglês
Publicado em: Springer Netherlands 2020
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Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC7524976/
https://ncbi.nlm.nih.gov/pubmed/32720036
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1007/s11302-020-09715-0
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