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Largazole is a Brain-Penetrant Class I HDAC Inhibitor with Extended Applicability to Glioblastoma and CNS Diseases

Largazole is a potent class I selective histone deacetylase (HDAC) inhibitor prodrug with anticancer activity against solid tumors in preclinical models. Largazole possesses in vitro activity against glioblastoma multiforme (GBM) cells and sufficiently crosses the blood-brain barrier based on measur...

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Bibliografski detalji
Izdano u:ACS Chem Neurosci
Glavni autori: Al-Awadhi, Fatma H., Salvador-Reyes, Lilibeth A., Elsadek, Lobna A., Ratnayake, Ranjala, Chen, Qi-Yin, Luesch, Hendrik
Format: Artigo
Jezik:Inglês
Izdano: 2020
Teme:
Online pristup:https://ncbi.nlm.nih.gov/pmc/articles/PMC7390227/
https://ncbi.nlm.nih.gov/pubmed/32559056
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acschemneuro.0c00093
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