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Largazole is a Brain-Penetrant Class I HDAC Inhibitor with Extended Applicability to Glioblastoma and CNS Diseases

Largazole is a potent class I selective histone deacetylase (HDAC) inhibitor prodrug with anticancer activity against solid tumors in preclinical models. Largazole possesses in vitro activity against glioblastoma multiforme (GBM) cells and sufficiently crosses the blood-brain barrier based on measur...

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Bibliografiska uppgifter
I publikationen:ACS Chem Neurosci
Huvudupphovsmän: Al-Awadhi, Fatma H., Salvador-Reyes, Lilibeth A., Elsadek, Lobna A., Ratnayake, Ranjala, Chen, Qi-Yin, Luesch, Hendrik
Materialtyp: Artigo
Språk:Inglês
Publicerad: 2020
Ämnen:
Länkar:https://ncbi.nlm.nih.gov/pmc/articles/PMC7390227/
https://ncbi.nlm.nih.gov/pubmed/32559056
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acschemneuro.0c00093
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