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Largazole: From Discovery to Broad-Spectrum Therapy

The cyclic depsipeptide largazole from a cyanobacterium of the genus Symploca is a marine natural product with novel chemical scaffold and potently inhibits class I histone deacetylases (HDACs). Largazole possesses highly differential growth-inhibitory activity, preferentially targeting transformed...

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Detalles Bibliográficos
Publicado en:Nat Prod Rep
Main Authors: Hong, Jiyong, Luesch, Hendrik
Formato: Artigo
Idioma:Inglês
Publicado: 2012
Assuntos:
Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC4777309/
https://ncbi.nlm.nih.gov/pubmed/22334030
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1039/c2np00066k
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