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Synthesis and Biological Evaluation of Largazole Zinc-Binding Group Analogs

Histone acetylation is an extensively investigated post-translational modification that plays an important role as an epigenetic regulator. It is controlled by histone acetyl transferases (HATs) and histone deacetylases (HDACs). The overexpression of HDACs and consequent hypoacetylation of histones...

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Publicat a:Bioorg Med Chem
Autors principals: Kim, Bumki, Ratnayake, Ranjala, Lee, Hyunji, Shi, Guqin, Zeller, Sabrina L., Li, Chenglong, Luesch, Hendrik, Hong, Jiyong
Format: Artigo
Idioma:Inglês
Publicat: 2017
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC5494147/
https://ncbi.nlm.nih.gov/pubmed/28416100
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmc.2017.03.071
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