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Synthesis and HDAC Inhibitory Activity of Largazole Analogs: Alteration of the Zinc-Binding Domain and Macrocyclic Scaffold

[Image: see text] Fourteen analogs of the marine natural product largazole have been prepared and assayed against HDACs 1,2, 3, and 6. Olefin cross-metathesis was used to efficiently access six variants of the side-chain zinc-binding domain, while adaptation of our previously reported modular synthe...

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Detalhes bibliográficos
Main Authors: Bowers, Albert A., West, Nathan, Newkirk, Tenaya L., Troutman-Youngman, Annie E., Schreiber, Stuart L., Wiest, Olaf, Bradner, James E., Williams, Robert M.
Formato: Artigo
Idioma:Inglês
Publicado em: 2009
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Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC2673910/
https://ncbi.nlm.nih.gov/pubmed/19239241
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/ol900078k
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