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Delineation of the molecular determinants of the unique allosteric binding site of the orphan nuclear receptor RORγt

Nuclear receptors (NRs) are high-interest targets in drug discovery because of their involvement in numerous biological processes and diseases. Classically, NRs are targeted via their hydrophobic, orthosteric pocket. Although successful, this approach comes with challenges, including off-target effe...

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Detalles Bibliográficos
Publicado en:J Biol Chem
Autores principales: Leijten-van de Gevel, Iris A., Brunsveld, Luc
Formato: Artigo
Lenguaje:Inglês
Publicado: American Society for Biochemistry and Molecular Biology 2020
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC7335795/
https://ncbi.nlm.nih.gov/pubmed/32439807
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1074/jbc.RA120.013581
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