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Targeted Protein Degradation in Antibacterial Drug Discovery?

Drug induced degradation of a target protein is a novel concept in drug discovery. Traditionally drugs modulate activity, as opposed to abundance, of their targets. Degradation inducing ligands act catalytically. Thus, one advantage of target degradation over the classical on-target mechanism is tha...

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Dettagli Bibliografici
Pubblicato in:Prog Biophys Mol Biol
Autori principali: Gopal, Pooja, Dick, Thomas
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2019
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC7145722/
https://ncbi.nlm.nih.gov/pubmed/31738980
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.pbiomolbio.2019.11.005
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