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Targeted Protein Degradation in Antibacterial Drug Discovery?

Drug induced degradation of a target protein is a novel concept in drug discovery. Traditionally drugs modulate activity, as opposed to abundance, of their targets. Degradation inducing ligands act catalytically. Thus, one advantage of target degradation over the classical on-target mechanism is tha...

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Kaydedildi:
Detaylı Bibliyografya
Yayımlandı:Prog Biophys Mol Biol
Asıl Yazarlar: Gopal, Pooja, Dick, Thomas
Materyal Türü: Artigo
Dil:Inglês
Baskı/Yayın Bilgisi: 2019
Konular:
Online Erişim:https://ncbi.nlm.nih.gov/pmc/articles/PMC7145722/
https://ncbi.nlm.nih.gov/pubmed/31738980
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.pbiomolbio.2019.11.005
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