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Targeted Protein Degradation: from Chemical Biology to Drug Discovery

Traditional pharmaceutical drug discovery is almost exclusively focused on directly controlling protein activity to cure diseases. Modulators of protein activity, especially inhibitors, are developed and applied at high concentration to achieve maximal effects. Thereby, reduced bioavailability and o...

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Detalhes bibliográficos
Publicado no:Cell Chem Biol
Main Authors: Cromm, Philipp M., Crews, Craig M.
Formato: Artigo
Idioma:Inglês
Publicado em: 2017
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC5610075/
https://ncbi.nlm.nih.gov/pubmed/28648379
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.chembiol.2017.05.024
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