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Evaluation of high-affinity phenyltetrahydroisoquinoline aldoximes, linked through anti-triazoles, as reactivators of phosphylated cholinesterases

Acetylcholinesterase (AChE) is a pivotal enzyme in neurotransmission. Its inhibition leads to cholinergic crises and could ultimately result in death. A related enzyme butyrylcholinesterase (BChE) may act in the CNS as a co-regulator in terminating nerve impulses and is a natural plasma scavenger up...

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Publicat a:Toxicol Lett
Autors principals: Hrvat, Nikolina Maček, Kalisiak, Jarosław, Šinko, Goran, Radić, Zoran, Sharpless, K. Barry, Taylor, Palmer, Kovarik, Zrinka
Format: Artigo
Idioma:Inglês
Publicat: 2019
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC7053431/
https://ncbi.nlm.nih.gov/pubmed/31863869
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.toxlet.2019.12.016
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