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Interaction Kinetics of Oximes with Native, Phosphylated and Aged Human Acetylcholinesterase

Oximes are commonly used nucleophilic reactivators of alkyl phosphorylated and alkyl methylphosphonylated acetylcholinesterase (AChE) and butyrylcholinesterase (BuChE). Covalent inhibition of these enzymes by organophosphate (OP) pesticides results typically in phosphorylated enzymes, while covalent...

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Gorde:
Xehetasun bibliografikoak
Egile Nagusiak: Radić, Zoran, Kalisiak, Jaroslaw, Fokin, Valery V., Sharpless, K. Barry, Taylor, Palmer
Formatua: Artigo
Hizkuntza:Inglês
Argitaratua: 2010
Gaiak:
Sarrera elektronikoa:https://ncbi.nlm.nih.gov/pmc/articles/PMC2912944/
https://ncbi.nlm.nih.gov/pubmed/20412789
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.cbi.2010.04.014
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