Loading...

Intracellular receptor modulation: Novel approach to target GPCRs

Recent crystal structures of multiple G protein-coupled receptors (GPCRs) have revealed a highly conserved intracellular pocket that can be used to modulate these receptors from the inside. This novel intracellular site partially overlaps with the G protein and β-arrestin binding site, providing a n...

Fuld beskrivelse

Na minha lista:
Bibliografiske detaljer
Udgivet i:Trends Pharmacol Sci
Main Authors: Ortiz Zacarías, Natalia V., Lenselink, Eelke B., IJzerman, Adriaan P., Handel, Tracy M., Heitman, Laura H.
Format: Artigo
Sprog:Inglês
Udgivet: 2018
Fag:
Online adgang:https://ncbi.nlm.nih.gov/pmc/articles/PMC7048003/
https://ncbi.nlm.nih.gov/pubmed/29653834
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.tips.2018.03.002
Tags: Tilføj Tag
Ingen Tags, Vær først til at tagge denne postø!