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Intracellular receptor modulation: Novel approach to target GPCRs

Recent crystal structures of multiple G protein-coupled receptors (GPCRs) have revealed a highly conserved intracellular pocket that can be used to modulate these receptors from the inside. This novel intracellular site partially overlaps with the G protein and β-arrestin binding site, providing a n...

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Dettagli Bibliografici
Pubblicato in:Trends Pharmacol Sci
Autori principali: Ortiz Zacarías, Natalia V., Lenselink, Eelke B., IJzerman, Adriaan P., Handel, Tracy M., Heitman, Laura H.
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2018
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC7048003/
https://ncbi.nlm.nih.gov/pubmed/29653834
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.tips.2018.03.002
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