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Preclinical studies reveal MLN4924 is a promising new retinoblastoma therapy

RB1 loss (RB1(null)) or MYCN amplification (MYCN(amp)) in fetal human retina causes retinoblastoma. SKP2 loss kills RB1(null) cells, but small molecule SKP2 inhibitors remain unexplored therapeutically. Whether SKP2 is synthetic lethal in MYCN(amp) retinoblastoma is unclear. SKP2 is the substrate re...

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Bibliografski detalji
Izdano u:Cell Death Discov
Glavni autori: Aubry, Arthur, Yu, Tao, Bremner, Rod
Format: Artigo
Jezik:Inglês
Izdano: Nature Publishing Group UK 2020
Teme:
Online pristup:https://ncbi.nlm.nih.gov/pmc/articles/PMC7026052/
https://ncbi.nlm.nih.gov/pubmed/32123578
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/s41420-020-0237-8
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