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Targeting dePARylation for cancer therapy

Poly(ADP-ribosyl)ation (PARylation) mediated by poly ADP-ribose polymerases (PARPs) plays a key role in DNA damage repair. Suppression of PARylation by PARP inhibitors impairs DNA damage repair and induces apoptosis of tumor cells with repair defects. Thus, PARP inhibitors have been approved by the...

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Publicat a:Cell Biosci
Autors principals: Kassab, Muzaffer Ahmad, Yu, Lily L., Yu, Xiaochun
Format: Artigo
Idioma:Inglês
Publicat: BioMed Central 2020
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC6988220/
https://ncbi.nlm.nih.gov/pubmed/32010441
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1186/s13578-020-0375-y
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