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Targeting dePARylation for cancer therapy
Poly(ADP-ribosyl)ation (PARylation) mediated by poly ADP-ribose polymerases (PARPs) plays a key role in DNA damage repair. Suppression of PARylation by PARP inhibitors impairs DNA damage repair and induces apoptosis of tumor cells with repair defects. Thus, PARP inhibitors have been approved by the...
Wedi'i Gadw mewn:
| Cyhoeddwyd yn: | Cell Biosci |
|---|---|
| Prif Awduron: | , , |
| Fformat: | Artigo |
| Iaith: | Inglês |
| Cyhoeddwyd: |
BioMed Central
2020
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| Pynciau: | |
| Mynediad Ar-lein: | https://ncbi.nlm.nih.gov/pmc/articles/PMC6988220/ https://ncbi.nlm.nih.gov/pubmed/32010441 https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1186/s13578-020-0375-y |
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