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Targeting dePARylation for cancer therapy

Poly(ADP-ribosyl)ation (PARylation) mediated by poly ADP-ribose polymerases (PARPs) plays a key role in DNA damage repair. Suppression of PARylation by PARP inhibitors impairs DNA damage repair and induces apoptosis of tumor cells with repair defects. Thus, PARP inhibitors have been approved by the...

Deskribapen osoa

Gorde:
Xehetasun bibliografikoak
Argitaratua izan da:Cell Biosci
Egile Nagusiak: Kassab, Muzaffer Ahmad, Yu, Lily L., Yu, Xiaochun
Formatua: Artigo
Hizkuntza:Inglês
Argitaratua: BioMed Central 2020
Gaiak:
Sarrera elektronikoa:https://ncbi.nlm.nih.gov/pmc/articles/PMC6988220/
https://ncbi.nlm.nih.gov/pubmed/32010441
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1186/s13578-020-0375-y
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