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Inhibition of hedgehog signaling by stereochemically defined des-triazole itraconazole analogues

Dysregulation of the hedgehog (Hh) signaling pathway is associated with cancer occurrence and development in various malignancies. Previous structure-activity relationships (SAR) studies have provided potent Itraconazole (ITZ) analogues as Hh pathway antagonists. To further expand on our SAR for the...

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Detalles Bibliográficos
Publicado en:Bioorg Med Chem Lett
Main Authors: Wen, Jiachen, Teske, Kelly A., Hadden, M. Kyle
Formato: Artigo
Idioma:Inglês
Publicado: 2019
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Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC6942223/
https://ncbi.nlm.nih.gov/pubmed/31761657
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmcl.2019.126794
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